journal article·2025-06-26

LumiCharge: Spherical Harmonic Convolutional Networks for Atomic Charge Prediction in Drug Discovery

Qun Su, Hui Zhang, Qiaolin Gou, Huiyong Sun, Meijing Fang, Xujun Zhang, Renling Hu, Yu Kang, Chang-Yu Hsieh, Jike Wang, Tingjun Hou

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Abstract

Atomic charge is crucial in drug design for analyzing reactive sites and interactions between ligands and targets. While quantum mechanical methods offer high accuracy, they are generally computationally costly. Conversely, empirical approaches, while computationally efficient, frequently suffer from lack of precision and generalizability. Recent a number of machine learning-based models have been developed for atomic charge predictions, but they struggle with accurately representing molecular structures and capturing the chemical environments affecting atomic charges, thus limiting their generalization and accuracy. To overcome these limitations, we propose LumiCharge, a novel atomic charge prediction framework that incorporates high-order spherical harmonics convolutions and explicitly models multibody interactions. In constructing this model, we employ a strategy that integrates both high- and low-order information, enhancing its geometric spatial perception capability, which is currently underexplored in the field. Benchmark evaluations demonstrate that LumiCharge outperforms state-of-the-art (SOTA) models by 30%-60% across diverse data sets. Additionally, in cross-scale experiments, LumiCharge demonstrates exceptional extrapolation capability and robustness across molecules of varying sizes, effectively overcoming the limitations imposed by molecular sizes. On an external halogen-containing test set, LumiCharge achieves an RMSE of 0.055e, meeting practical application requirements. Finally, a case study of virtual screening for the androgen receptor (AR) target further validates its outstanding accuracy compared to the OPLS3e force field and other deep learning (DL)-based baseline models, highlighting its exceptional generalization capacity and practical utility in real-world scenarios.
Source: openalex_inverted_index · Quality: baseline

Research context

OpenAlex topics: Computational Drug Discovery Methods · thermodynamics and calorimetric analyses · Mass Spectrometry Techniques and Applications

SciVX discovery tags are terminology-based. OpenAlex topics are source-provided classifications.

Affiliations

College of Pharmaceutical Sciences

Zhejiang University

Faculty of Applied Sciences

Macao Polytechnic University

Department of Medicinal Chemistry

China Pharmaceutical University

Zhejiang Provincial Key Laboratory for Intelligent Drug Discovery and Development

Funding

National Key Research and Development Program of China · National Natural Science Foundation of China

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